| US 7,462,735 B2 | ||
| Amino acid diamides in non α position which are useful as adjuvants for administration of biological active agents | ||
| Jean Sarkis Mardiguian, Madrid (Spain) | ||
| Assigned to Laboratorios Farmaceuticos Rovi, S.A., Madrid (Spain) | ||
| Appl. No. 10/563,994 PCT Filed Jul. 23, 2004, PCT No. PCT/ES2004/000346 § 371(c)(1), (2), (4) Date Jul. 14, 2006, PCT Pub. No. WO2005/012230, PCT Pub. Date Feb. 10, 2005. |
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| Claims priority of application No. 200301781 (ES), filed on Jul. 28, 2003. | ||
| Prior Publication US 2007/0191302 A1, Aug. 16, 2007 | ||
| Int. Cl. C07C 229/00 (2006.01); A61K 31/715 (2006.01); A61K 31/727 (2006.01); A61K 31/195 (2006.01) | ||
| U.S. Cl. 562—450 [514/54; 514/56; 514/563] | 15 Claims |
1. Amino acid diamides in non-α position of formula (1)
 R1 is selected from the group consisting of halogen, NO2, OH, OCH3 and a combination thereof; and
R2 is selected from the group consisting of H, alkyl, halogen, NO2, OH, and OCH3.
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