| US 7,456,133 B2 | ||
| Substituted arylketones | ||
| Stefan Herrmann, Langenfeld (Germany); Dorothee Hoischen, Dusseldorf (Germany); Kristian Kather, Lagenfeld (Germany); Klaus-Helmut Muller, Dusseldorf (Germany); Otto Schallner, Monheim (Germany); Hans-Georg Schwarz, Lagenfeld (Germany); Mark Wilhelm Drewes, Langenfeld (Germany); Peter Dahmen, Neuss (Germany); Dieter Feucht, Monheim (Germany); and Rolf Pontzen, Leichlingen (Germany) | ||
| Assigned to Bayer CropScience AG, Monheim (Germany) | ||
| Filed on Jul. 10, 2006, as Appl. No. 11/483,892. | ||
| Application 11/483892 is a division of application No. 10/477031, granted, now 7,112,554, filed on Sep. 26, 2006, previously published as PCT/EP02/04701, filed on Apr. 29, 2002. | ||
| Claims priority of application No. 101 22 445 (DE), filed on May 09, 2001; and application No. 101 36 449 (DE), filed on Jul. 26, 2001. | ||
| Prior Publication US 2006/0252647 A1, Nov. 09, 2006 | ||
| Int. Cl. A01N 43/80 (2006.01); A01N 43/56 (2006.01); C07D 261/08 (2006.01); C07D 231/20 (2006.01) | ||
| U.S. Cl. 504—271 [504/280; 548/248; 548/369.4] | 8 Claims |
1. A compound of the Formula (I)
![]() A1 represents a single bond or represents O, S, SO, SO2,
A2 represents alkanediyl (alkylene), alkenediyl or alkinediyl,
Q represents O (oxygen) or S (sulphur),
R1 represents hydrogen or represents in each case optionally substituted alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl,
alkylamino, dialkylamino, alkenyl, alkinyl, cycloalkyl, cycloalkylalkyl, aryl or arylalkyl, or represents the grouping —C(Q)-R2,
R2 represents hydrogen, amino, cyanoamino, nitroamino, hydroxyamino, hydrazino, or represents in each case optionally substituted
alkyl, alkylcarbonyl, alkoxy, alkoxycarbonyl, alkylthio, alkylamino, dialkylamino, alkoxyamino, N-alkyl-alkoxyamino, alkylhydrazino,
dialkylhydrazino, alkenyl, alkenyloxy, alkenylamino, alkenyloxyamino, alkinyl, alkinyloxy, alkinylamino, cycloalkyl, cycloalkyloxy,
cycloalkylamino, cycloalkylalkyl, cycloalkylalkoxy, cycloalkylalkylamino, aryl, arylcarbonyl, aryloxy, aryloxycarbonyl, arylthio,
arylamino, arylhydrazino, arylalkyl, arylalkoxy, arylalkylthio, arylalkylamino, heterocyclyl, heterocyclyloxy, heterocyclylthio,
heterocyclylamino, heterocyclylalkyl, heterocyclylalkoxy, heterocyclylalkylthio or heterocyclylalkylamino,
X represents hydrogen, nitro, cyano, carboxyl, carbamoyl, thiocarbamoyl, halogen, or represents in each case optionally substituted
alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl, alkylamino, dialkylamino or dialkylaminosulphonyl,
Y represents hydrogen, nitro, cyano, carboxyl, carbamoyl, thiocarbamoyl, halogen, or represents in each case optionally substituted
alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl, alkylamino, dialkylamino or dialkylaminosulphonyl, and
Z represents one of the groupings below
![]() m represents the numbers 0 to 6,
R3 represents hydrogen, halogen or represents in each case optionally substituted alkyl, alkylthio or aryl, or—if m represents
2—optionally also together with a second radical R3 represents oxygen or alkanediyl (alkylene),
R4 represents hydroxyl, formyloxy, halogen, or represents in each case optionally substituted alkoxy, alkylthio, alkylsulphinyl,
alkylsulphonyl, alkylcarbonyloxy, alkoxycarbonyloxy, alkylaminocarbonyloxy, alkylsulphonyloxy, alkenyloxy, alkinyloxy, aryloxy,
arylthio, arylsulphinyl, arylsulphonyl, arylcarbonyloxy, arylcarbonylalkoxy, arylsulphonyloxy, arylalkoxy, arylalkylthio,
arylalkylsulphinyl or arylalkylsulphonyl,
R5 represents hydrogen, cyano, carbamoyl, thiocarbamoyl, halogen, or represents in each case optionally substituted alkyl, alkoxy,
alkylthio, alkylsulphinyl, alkylsulphonyl, alkoxycarbonyl or cycloalkyl,
R6 represents hydrogen or represents in each case optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkylalkyl,
aryl or arylalkyl,
R7 represents hydroxyl, formyloxy, or represents in each case optionally substituted alkoxy, alkylcarbonyloxy, alkoxycarbonyloxy,
alkylaminocarbonyloxy, alkylsulphonyloxy, alkenyloxy, alkinyloxy, arylalkoxy, arylcarbonyloxy, arylcarbonylalkoxy or arylsulphonyloxy,
R8 represents hydrogen, cyano, carbamoyl, thiocarbamoyl, halogen, or represents in each case optionally substituted alkyl, alkylcarbonyl,
alkoxy, alkoxycarbonyl, alkylthio, alkylsulphinyl or alkylsulphonyl,
R9 represents hydrogen or represents in each case optionally substituted alkyl or cycloalkyl,
R10 represents hydrogen or represents in each case optionally substituted alkyl or cycloalkyl, and
R11 represents hydrogen, cyano, carbamoyl, halogen, or represents in each case optionally substituted alkyl, alkoxy, alkoxycarbonyl,
alkylthio, alkylsulphinyl or alkylsulphonyl
with the proviso that when Q is oxygen, R2 is not cyclopropyl and Z is not
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