US 7,576,202 B2
Tritium-traced saxitoxin dihydrochloride and method for the production thereof
Nikolay Fedorovich Myasoedov, Moscow (Russian Federation); Valery Pavlovich Shevchenko, Moscow (Russian Federation); Igor Yulianovich Nagaev, Moskovskaya obl. (Russian Federation); and Alexander Susan, Leawood, Kans. (US)
Assigned to Institut Molekulyarnoi Genetiki Rossiiskoi Akademh Nauk (IMG RAN), (Russian Federation)
Appl. No. 11/722,926
PCT Filed Dec. 27, 2005, PCT No. PCT/RU2005/000672
§ 371(c)(1), (2), (4) Date Nov. 01, 2007,
PCT Pub. No. WO2006/071138, PCT Pub. Date Jul. 06, 2006.
Claims priority of application No. 2004138131 (RU), filed on Dec. 27, 2004.
Prior Publication US 2008/0091013 A1, Apr. 17, 2008
Int. Cl. C07D 491/00 (2006.01)
U.S. Cl. 544—251 17 Claims
 
1. A tritium-traced saxitoxin dihydrochloride of formula (I)

OG Complex Work Unit Drawing
having a radioactivity of 15-31 Ci/mmol.